BCL6 inhibitor 7

CAS No. 2097518-46-0

BCL6 inhibitor 7( BCL6-IN-7 | BCL6 IN 7 | BCL6IN7 | BCL6 inhibitor-7 )

Catalog No. M13307 CAS No. 2097518-46-0

A potent BCL6 protein-protein interaction inhibitor with Kd of 78 nM; exhibits an efficacy in cell-free and cellular PPI assays.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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Biological Information

  • Product Name
    BCL6 inhibitor 7
  • Note
    Research use only, not for human use.
  • Brief Description
    A potent BCL6 protein-protein interaction inhibitor with Kd of 78 nM; exhibits an efficacy in cell-free and cellular PPI assays.
  • Description
    A potent BCL6 protein-protein interaction inhibitor with Kd of 78 nM; exhibits an efficacy in cell-free and cellular PPI assays (ELISA IC50= 480 nM, M2H IC50= 8.6 uM).
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    BCL6-IN-7 | BCL6 IN 7 | BCL6IN7 | BCL6 inhibitor-7
  • Pathway
    Angiogenesis
  • Target
    Bcl-2
  • Recptor
    Bcl-2
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    2097518-46-0
  • Formula Weight
    366.809
  • Molecular Formula
    C18H15ClN6O
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 5 mg/mL (13.63 mM)
  • SMILES
    O=C1NC2=C(C=C(NC3=NC(NCC4=CC=CN=C4)=NC=C3Cl)C=C2)C1
  • Chemical Name
    5-((5-Chloro-2-((pyridin-3-ylmethyl)amino)pyrimidin-4-yl)-amino)-1,3-dihydro-2H-indol-2-one

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Kamada Y, et al. J Med Chem. 2017 May 25;60(10):4358-4368.
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